光亲和标记
DNA
小分子
化学
化学生物学
药物发现
组合化学
计算生物学
生物化学
结构生物学
生物物理学
结合位点
生物
作者
Gang Li,Ying Liu,Yu Liu,Li Chen,Siyu Wu,Yang Liu,Xiaoyu Li
标识
DOI:10.1002/anie.201302161
摘要
DNA-templated affinity labeling: Accurate characterization of small-molecule (SM)–protein interactions is one of the most important but also very challenging tasks in chemical biology and drug discovery. A novel method named DNA-programmed photoaffinity labeling is reported. The introduction of DNA encoding and template effect enable multiplexed protein labeling by multiple probes.
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