喹啉酮
抗真菌
广谱
化学
药理学
组合化学
生物
微生物学
作者
Dan He,Menglei Wang,Siyu Zhao,Yisong Shu,Honglian Zeng,Cheng Xiao,Cheng Lü,Yuanyan Liu
出处
期刊:Fitoterapia
[Elsevier]
日期:2017-06-01
卷期号:119: 136-149
被引量:88
标识
DOI:10.1016/j.fitote.2017.05.001
摘要
Quinazolinones belong to a family of heterocyclic nitrogen compounds that have attracted increasing interest because of their broad spectrum of biological functions. This review describes three types of natural quinazolinones and their synthesized derivatives and summarizes their various pharmacological activities, including antifungal, anti-tumor, anti-malaria, anticonvulsant, anti-microbial, anti-inflammatory and antihyperlipidemic activities. In addition, structure-activity relationships of quinazolinone derivatives are also reviewed.
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