化学
抗真菌
双功能
酶抑制剂
药理学
组合化学
生物化学
酶
微生物学
医学
生物
催化作用
作者
Haibo Liu,Shuai Yu,Yan‐Qin He,Shiying Zhang,Min Liu,Jun Han,Bin Sun
标识
DOI:10.1021/acs.jmedchem.4c01057
摘要
Fungal infections maintain a close relation with the body's immune function. In this study, three series of benzazole compounds were designed as dual-target (PD-L1/CYP51) inhibitors using the skeleton splicing approach; their molecular structures were synthesized and evaluated accordingly. Among them, the compounds
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