CYP2C8
细胞色素P450
药物代谢
化学
药理学
药品
新陈代谢
药物遗传学
生物化学
医学
CYP2C9
基因
基因型
作者
Xiaoping Liu,Fangfang Zhong,Xiangshi Tan
标识
DOI:10.2174/15680266113136660157
摘要
CYP 2C8, which carries out the oxidative metabolism of at least 5% of clinical drugs, has attracted increasing attention in recent years. New drugs (substances), inducers and inhibitors of CYP 2C8 have been developed and the drug metabolism has been investigated to understand the clinical role of CYP2C8. The cases of CYP2C8 genetic polymorphisms linked to diseases have increased and have been investigated. Herein, important progress in these areas has been reviewed with an emphasis on drug metabolism. Polymorphisms, diseases related to CYP2C8, some important drugs (substances) and inhibitors are reviewed and discussed.
科研通智能强力驱动
Strongly Powered by AbleSci AI