化学
树皮(声音)
胰脂肪酶
植物化学
阳性对照
桑科
立体化学
脂肪酶
IC50型
传统医学
体外
有机化学
生物化学
酶
物理
医学
声学
作者
Manh Tuan Ha,Manh Hung Tran,Kim Jeong Ah,Kyung-Jin Jo,Jae-Wang Kim,Wook Dong Kim,Woo Jae Cheon,Mi Hee Woo,Sung Ho Ryu,Byung Sun Min
标识
DOI:10.1016/j.bmcl.2016.04.066
摘要
Detailed phytochemical investigation from the root bark of Morus alba resulted in the isolation of eleven new compounds, including seven 2-arylbenzofuran derivatives (morusalfurans A-G), three flavonoids (morusalnols A-C), and one geranylated stilbene (morusibene A), as well as 22 known compounds. The structures of the identified compounds were elucidated based on a comprehensive analysis of spectroscopic data and Mosher's method. Compounds 2, 3, 6-8, 11, 23, 24, and 29 showed potent inhibition of PL in comparison with the positive control treatment (orlistat, IC50=0.012μM), with IC50 values ranging from 0.09 to 0.92μM.
科研通智能强力驱动
Strongly Powered by AbleSci AI