计算生物学
化学
癌细胞
生物
细胞生物学
生物化学
癌症
遗传学
作者
Lingsha Zhou,Cai-Guang Yang
出处
期刊:Structure
[Elsevier]
日期:2023-02-01
卷期号:31 (2): 125-127
被引量:1
标识
DOI:10.1016/j.str.2023.01.002
摘要
In this issue of Structure, Mabanglo et al. characterize five ClpP agonists termed TRs. The co-crystal structures reveal more robust shape and charge complementarities than the anti-cancer agent ONC201. These novel compounds are of potential therapeutic interest because they enhance ClpP proteolytic activity and have an inhibitory effect on tumor cell growth.
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