血脑屏障
运输机
药物输送
药物输送到大脑
药理学
神经药理学
药品
神经科学
医学
生物
化学
中枢神经系统
生物化学
有机化学
基因
作者
Patrick T. Ronaldson,Thomas P. Davis
标识
DOI:10.1080/17425247.2024.2306138
摘要
Introduction Successful neuropharmacology requires optimization of CNS drug delivery and, by extension, free drug concentrations at brain molecular targets. Detailed assessment of blood-brain barrier (BBB) physiological characteristics is necessary to achieve this goal. The 'next frontier' in CNS drug delivery is targeting BBB uptake transporters, an approach that requires evaluation of brain endothelial cell transport processes so that effective drug accumulation and improved therapeutic efficacy can occur.
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