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朴素觅风
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40 积分
2023-08-01 加入
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Discovery of orally bioavailable ALK PROTACs based Ceritinib against ALK positive cancers
1小时前
待确认
Dual-ligand PROTACS mediate superior target protein degradation in vitro and therapeutic efficacy in vivo
2小时前
已完结
Discovery of novel 20S proteasome subunit β5 PROTAC degraders as potential therapeutics for pharyngeal carcinoma and Bortezomib-resistant multiple myeloma
12天前
已完结
Discovery of highly efficient CRBN-recruiting HPK1-PROTAC as a potential chemical tool for investigation of scaffolding roles in TCR signaling
1个月前
已完结
PROTACs: Novel tools for improving immunotherapy in cancer
1个月前
已完结
One-Pot Synthesis of Cereblon Proteolysis Targeting Chimeras via Photoinduced C(sp2)–C(sp3) Cross Coupling and Amide Formation for Proteolysis Targeting Chimera Library Synthesis
1个月前
已完结
Selective degradation of histone deacetylase 8 mediated by a proteolysis targeting chimera (PROTAC)
1个月前
已完结
Discovery of pomalidomide-based PROTACs for selective degradation of histone deacetylase 8
1个月前
已完结
Discovery of FLT3-targeting PROTACs with potent antiproliferative activity against acute myeloid leukemia cells harboring FLT3 mutations
1个月前
已完结
Discovery of FLT3-targeting PROTACs with potent antiproliferative activity against acute myeloid leukemia cells harboring FLT3 mutations
1个月前
已完结
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2个月前
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