伊萨丁
化学
体内
体外
生物化学
组合化学
药理学
计算生物学
有机化学
生物技术
生物
作者
Shital Patil,Shankar G. Alegaon,Shankar Gharge,Shriram D. Ranade,Nayeem A. Khatib
标识
DOI:10.1016/j.bioorg.2024.107783
摘要
In the pursuit of novel antidiabetic agents, a series of isatin-thiazole derivatives (7a-7j) were synthesized and characterized using a range of spectroscopic techniques. The enzyme inhibitory activities of the target analogues were assessed using both in vitro and in vivo assays. The tested compounds 7a-7j demonstrated In vitro inhibitory potential against α-glucosidase, as indicated by their IC
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