咖啡酸苯乙酯
血红素加氧酶
咖啡酸
氧化应激
诱导剂
血红素
细胞保护
化学
生物化学
氧化磷酸化
加氧酶
酶
药理学
抗氧化剂
生物
基因
作者
Valeria Pittalà,Luca Vanella,Loredana Salerno,Claudia Di Giacomo,Rosaria Acquaviva,Marco Raffaele,Giuseppe Romeo,Maria Modica,Orazio Prezzavento,Valeria Sorrenti
标识
DOI:10.2174/1381612823666170210151411
摘要
Background:Heme Oxygenase-1 (HO-1) is a metabolic enzyme strongly involved in processes including cytoprotection, modulation of inflammatory response, anti-oxidative functions, regulation of cellular proliferation, angiogenesis, cardiovascular homeostasis, and immuno-modulation. HO-1 induction and/or activation is able to counterbalance, at least in part, oxidative stress and inflammation. For this reason, HO-1 can be regarded as an attractive target to ameliorate different stress-related pathologies. Caffeic acid phenethyl ester, a natural polyphenolic compound, behaves as HO-1 inducer and possesses a plethora of beneficial effects under oxidative stress conditions. Keywords: Heme oxygenase, HO-1 inducers, caffeic acid phenethyl ester, ROS, human MSCs, VP961.
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