绞股蓝
细胞凋亡
生物利用度
药理学
传统医学
癌症研究
化学
医学
生物化学
萃取(化学)
色谱法
作者
Kaijun Li,Chao Ma,Haoyu Li,Sooranna Dev,Jianfeng He,Xiaosheng Qu
标识
DOI:10.2174/1568026619666191114104718
摘要
: Gynostemma pentaphyllum (Thunb.) Makino (GpM) and its derivatives, especially gypenosides (Gyps), are widely used as safe and convenient natural herbal drugs for the treatment of many diseases for a long time, and Gyps have different oral bioavailability (OB) values and low ability to cross the blood-brain barrier (BBB). The effects of GpM and isolates on fibrosis, inflammation, oxidation, proliferation and migration are proved. GpM shows bidirectional regulation effect on proliferation, oxidation and apoptosis in tumor and non-tumor cells. GpM and its extractions can resist proliferation, activate oxidation and apoptosis in tumor cells and have opposite effects on non-tumor cells. We succinctly present some current views of medicinal value and potential therapeutic mechanisms of GpM and its derivatives.
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