化学
卡铂
细胞毒性
杯芳烃
铂金
组合化学
细胞培养
细胞毒性T细胞
IC50型
立体化学
体外
顺铂
生物化学
有机化学
化疗
内科学
分子
催化作用
生物
医学
遗传学
作者
Fazel Nasuhi Pur,Karim Akbari Dilmaghani
标识
DOI:10.1080/00958972.2014.890718
摘要
A functionalized calixarene with four platinum(II) centers was synthesized as a potential anticancer agent. The colorimetric cytotoxicity tests showed that it has amplified activity with respect to carboplatin against three different human carcinoma (non-small-cell lung, hepatocellular, and breast cancer) cell lines. It was most cytotoxic against the lung cancer cell line (IC50 = 2.6 μM).
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