5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]- [1,4]benzodiazepin-10(11H)-ylcarbonyl)-3- chlorophenyl]benzamide (VPA-985): An Orally Active Arginine Vasopressin Antagonist with Selectivity for V2Receptors

ADVERTISEMENT RETURN TO ISSUEPREVLetterNEXT5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]- [1,4]benzodiazepin-10(11H)-ylcarbonyl)-3- chlorophenyl]benzamide (VPA-985): An Orally Active Arginine Vasopressin Antagonist with Selectivity for V2 ReceptorsJ. Donald Albright, Marvin F. Reich, Efren G. Delos Santos, John P. Dusza, Fuk-Wah Sum, Aranapakam M. Venkatesan, Joseph Coupet, Peter S. Chan, Xun Ru, Hossein Mazandarani, and Trina BaileyView Author Information Wyeth-Ayerst Research, Pearl River, New York 10965, and Wyeth-Ayerst Research, Princeton, New Jersey 08543-8000 Cite this: J. Med. Chem. 1998, 41, 14, 2442–2444Publication Date (Web):June 16, 1998Publication History Received23 March 1998Published online16 June 1998Published inissue 1 July 1998https://pubs.acs.org/doi/10.1021/jm980179chttps://doi.org/10.1021/jm980179crapid-communicationACS PublicationsCopyright © 1998 American Chemical SocietyRequest reuse permissionsArticle Views1035Altmetric-Citations125LEARN ABOUT THESE METRICSArticle Views are the COUNTER-compliant sum of full text article downloads since November 2008 (both PDF and HTML) across all institutions and individuals. These metrics are regularly updated to reflect usage leading up to the last few days.Citations are the number of other articles citing this article, calculated by Crossref and updated daily. Find more information about Crossref citation counts.The Altmetric Attention Score is a quantitative measure of the attention that a research article has received online. Clicking on the donut icon will load a page at altmetric.com with additional details about the score and the social media presence for the given article. Find more information on the Altmetric Attention Score and how the score is calculated. Share Add toView InAdd Full Text with ReferenceAdd Description ExportRISCitationCitation and abstractCitation and referencesMore Options Share onFacebookTwitterWechatLinked InRedditEmail Other access optionsGet e-AlertscloseSupporting Info (1)»Supporting Information Supporting Information SUBJECTS:Antagonists,Receptors,Rodent models,Screening assays,Selectivity Get e-Alerts